国立医薬品食品衛生研究所 |
National Institute of Health Sciences |
生物薬品部 |
Division of Biological Chemistry and Biologicals |
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【rINN】teprotumumab (List 63, 2010, Vol.24, No. 1, p77)
【pINN】teprotumumab (List 101, 2009, Vol.23, No. 2, p170)
【解説(和訳)】
IgG1κ, 抗ヒトインスリン様成長因子1受容体 (IGF1R, IGF-1R, IGF-1 receptor, CD221), ヒトモノクローナル抗体;
抗腫瘍薬.
H鎖 (γ1鎖,1-448) [Homo sapiens VH (IGHV3-33*01 (91.80%) -(IGHD)-IGHJ2*01)
[8.8.11] (1-118) -IGHG1*01 (119-448)], (221-215')].
L鎖(κ鎖,1'-215') [Homo sapiens VKAPPA (IGKV3-11*01 (97.90%) -IGKJ1*01) [6.3.10]
(1'-108') -IGKC*01 (109'-215')].
ジスルフィド結合の位置: 221-215', 227-227'', 230-230''
糖鎖付加位置 298, 298''
【分子式】C6476H10012N1748O2000S40
【CAS番号】89957-37-9
【JAN】未収載
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